Compound ID | NCGC00185684 | NCGC00184846 |
---|---|---|
Code name | NCGC84 | SHA68 |
Structure | ||
IC50 - cAMP | 22.1 ± 1.9 | 208.3 ± 36.3 |
IC50 - Ca2+ | 36.5 ± 6.4 | 569.6 ± 130.3 |
IC50 - ERK-phospho | 9.3 ± 11.5 | 15.8 ± 2.7 |
IC50 - binding (95% CI) | 5.0 (3.88–6.42) | 9.5 (53.2–73.4) |
pA2 (95% CI) | 8.98 (9.03–8.94) | 8.16 (8.25–8.08) |
Schild slope | 1.03 ± 0.01 | 1.00 ± 0.03 |